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CYP2B6 is An important CYP enzyme involved in the metabolism of S-methadone and also to an extent, R-methadone. The expression of CYP2B6Benzodiazepines: May enrich the CNS depressant effect of Methadone. Management: Clinicians ought to generally steer clear of concurrent utilization of methadone and benzodiazepines when probable; any blended use sh